{"product_id":"pt-141-10mg-vial","title":"PT-141 10mg vial","description":"\u003cp data-start=\"87\" data-end=\"482\"\u003e\u003cstrong\u003e\u003cstrong data-start=\"377\" data-end=\"392\"\u003e\u003cspan style=\"color: rgb(255, 42, 0);\"\u003e                                             \u003cspan style=\"text-decoration: underline;\"\u003eNOT \u003c\/span\u003e\u003c\/span\u003e\u003cspan style=\"text-decoration: underline;\"\u003e\u003cspan style=\"color: rgb(255, 42, 0); text-decoration: underline;\"\u003eFOR HUMAN CONSUMPTION\u003c\/span\u003e\u003c\/span\u003e\u003c\/strong\u003e\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp data-start=\"87\" data-end=\"482\"\u003e\u003cstrong\u003ePT-141\u003c\/strong\u003e, also known as \u003cstrong data-start=\"109\" data-end=\"126\"\u003eBremelanotide\u003c\/strong\u003e, is a synthetic peptide that acts as a melanocortin receptor agonist. It was initially developed as a tanning agent but was later found to have significant effects on sexual arousal and dysfunction. Unlike PDE5 inhibitors like \u003cstrong data-start=\"354\" data-end=\"364\"\u003eViagra\u003c\/strong\u003e or \u003cstrong data-start=\"368\" data-end=\"378\"\u003eCialis\u003c\/strong\u003e, PT-141 works through the \u003cstrong data-start=\"405\" data-end=\"437\"\u003ecentral nervous system (CNS)\u003c\/strong\u003e rather than directly affecting blood flow.\u003c\/p\u003e\n\u003ch4 data-start=\"484\" data-end=\"514\"\u003e\u003cstrong data-start=\"489\" data-end=\"512\"\u003eMechanism of Action\u003c\/strong\u003e\u003c\/h4\u003e\n\u003cp data-start=\"515\" data-end=\"831\"\u003ePT-141 primarily targets \u003cstrong data-start=\"540\" data-end=\"582\"\u003emelanocortin receptors (MC3R and MC4R)\u003c\/strong\u003e in the brain, which are involved in sexual arousal. By stimulating these receptors, it enhances libido and sexual response \u003cstrong data-start=\"706\" data-end=\"748\"\u003eindependently of nitric oxide pathways\u003c\/strong\u003e, making it effective even for individuals who do not respond to PDE5 inhibitors.\u003c\/p\u003e\n\u003ch4 data-start=\"833\" data-end=\"861\"\u003e\u003cstrong data-start=\"838\" data-end=\"859\"\u003eUses and Benefits\u003c\/strong\u003e\u003c\/h4\u003e\n\u003col data-start=\"862\" data-end=\"1580\"\u003e\n\u003cli data-start=\"862\" data-end=\"1118\"\u003e\n\u003cp data-start=\"865\" data-end=\"902\"\u003e\u003cstrong data-start=\"865\" data-end=\"900\"\u003eTreatment of Sexual Dysfunction\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul data-start=\"906\" data-end=\"1118\"\u003e\n\u003cli data-start=\"906\" data-end=\"1028\"\u003e\n\u003cstrong data-start=\"908\" data-end=\"969\"\u003eFDA-approved for HSDD (Hypoactive Sexual Desire Disorder)\u003c\/strong\u003e in premenopausal women under the brand name \u003cstrong data-start=\"1014\" data-end=\"1025\"\u003eVyleesi\u003c\/strong\u003e.\u003c\/li\u003e\n\u003cli data-start=\"1032\" data-end=\"1114\"\u003eMay be used \u003cstrong data-start=\"1046\" data-end=\"1089\"\u003eoff-label for erectile dysfunction (ED)\u003c\/strong\u003e and low libido in men.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"1119\" data-end=\"1346\"\u003e\n\u003cp data-start=\"1122\" data-end=\"1161\"\u003e\u003cstrong data-start=\"1122\" data-end=\"1159\"\u003ePotential Performance Enhancement\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul data-start=\"1165\" data-end=\"1346\"\u003e\n\u003cli data-start=\"1165\" data-end=\"1247\"\u003eIncreases \u003cstrong data-start=\"1177\" data-end=\"1222\"\u003esexual desire, arousal, and response time\u003c\/strong\u003e in both men and women.\u003c\/li\u003e\n\u003cli data-start=\"1251\" data-end=\"1346\"\u003eCan improve \u003cstrong data-start=\"1265\" data-end=\"1280\"\u003espontaneity\u003c\/strong\u003e in sexual activity, unlike PDE5 inhibitors that require timing.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"1348\" data-end=\"1580\"\u003e\n\u003cp data-start=\"1351\" data-end=\"1393\"\u003e\u003cstrong data-start=\"1351\" data-end=\"1374\"\u003ePossible Other Uses\u003c\/strong\u003e (Under Research)\u003c\/p\u003e\n\u003cul data-start=\"1397\" data-end=\"1580\"\u003e\n\u003cli data-start=\"1397\" data-end=\"1463\"\u003ePotential appetite suppression and weight regulation benefits.\u003c\/li\u003e\n\u003cli data-start=\"1467\" data-end=\"1580\"\u003eMay play a role in \u003cstrong data-start=\"1488\" data-end=\"1536\"\u003epain management and immune system regulation\u003c\/strong\u003e due to melanocortin receptor involvement.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003c\/li\u003e\n\u003c\/ol\u003e\n\u003ch4 data-start=\"1582\" data-end=\"1618\"\u003e\u003cstrong data-start=\"1587\" data-end=\"1616\"\u003eDosage and Administration\u003c\/strong\u003e\u003c\/h4\u003e\n\u003cul data-start=\"1619\" data-end=\"1896\"\u003e\n\u003cli data-start=\"1619\" data-end=\"1702\"\u003eTypically administered as a \u003cstrong data-start=\"1649\" data-end=\"1675\"\u003esubcutaneous injection\u003c\/strong\u003e in the abdomen or thigh.\u003c\/li\u003e\n\u003cli data-start=\"1703\" data-end=\"1811\"\u003e\n\u003cstrong data-start=\"1705\" data-end=\"1723\"\u003eStandard dose:\u003c\/strong\u003e 1.75 mg for HSDD in women (self-injected at least 45 minutes before sexual activity).\u003c\/li\u003e\n\u003cli data-start=\"1812\" data-end=\"1896\"\u003eEffects can last \u003cstrong data-start=\"1831\" data-end=\"1848\"\u003e6 to 12 hours\u003c\/strong\u003e, with residual effects up to \u003cstrong data-start=\"1878\" data-end=\"1893\"\u003e24-48 hours\u003c\/strong\u003e.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003ch4 data-start=\"1898\" data-end=\"1921\"\u003e\u003cstrong data-start=\"1903\" data-end=\"1919\"\u003eSide Effects\u003c\/strong\u003e\u003c\/h4\u003e\n\u003cul data-start=\"1922\" data-end=\"2197\"\u003e\n\u003cli data-start=\"1922\" data-end=\"1991\"\u003e\n\u003cstrong data-start=\"1924\" data-end=\"1935\"\u003eCommon:\u003c\/strong\u003e Nausea, flushing, headache, injection site reactions.\u003c\/li\u003e\n\u003cli data-start=\"1992\" data-end=\"2086\"\u003e\n\u003cstrong data-start=\"1994\" data-end=\"2010\"\u003eLess Common:\u003c\/strong\u003e Increased blood pressure, darkening of skin (hyperpigmentation), yawning.\u003c\/li\u003e\n\u003cli data-start=\"2087\" data-end=\"2197\"\u003e\n\u003cstrong data-start=\"2089\" data-end=\"2110\"\u003eRare but Serious:\u003c\/strong\u003e Cardiovascular risks (caution in individuals with hypertension or heart conditions).\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003ch4 data-start=\"2199\" data-end=\"2239\"\u003e\u003cstrong data-start=\"2204\" data-end=\"2237\"\u003eComparison to PDE5 Inhibitors\u003c\/strong\u003e\u003c\/h4\u003e\n\u003cdiv class=\"overflow-x-auto contain-inline-size\"\u003e\n\u003ctable data-start=\"2240\" data-end=\"2828\"\u003e\n\u003cthead data-start=\"2240\" data-end=\"2319\"\u003e\n\u003ctr data-start=\"2240\" data-end=\"2319\"\u003e\n\u003cth data-start=\"2240\" data-end=\"2258\"\u003eFeature\u003c\/th\u003e\n\u003cth data-start=\"2258\" data-end=\"2283\"\u003ePT-141 (Bremelanotide)\u003c\/th\u003e\n\u003cth data-start=\"2283\" data-end=\"2319\"\u003ePDE5 Inhibitors (Viagra, Cialis)\u003c\/th\u003e\n\u003c\/tr\u003e\n\u003c\/thead\u003e\n\u003ctbody data-start=\"2389\" data-end=\"2828\"\u003e\n\u003ctr data-start=\"2389\" data-end=\"2471\"\u003e\n\u003ctd\u003e\u003cstrong data-start=\"2391\" data-end=\"2409\"\u003eMode of Action\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd\u003eCentral nervous system\u003c\/td\u003e\n\u003ctd\u003ePeripheral vascular (blood flow)\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"2472\" data-end=\"2553\"\u003e\n\u003ctd\u003e\u003cstrong data-start=\"2474\" data-end=\"2494\"\u003eEffect on Libido\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd\u003eDirect increase in desire\u003c\/td\u003e\n\u003ctd\u003eNo effect on libido itself\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"2554\" data-end=\"2634\"\u003e\n\u003ctd\u003e\u003cstrong data-start=\"2556\" data-end=\"2570\"\u003eOnset Time\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd\u003e30-60 minutes\u003c\/td\u003e\n\u003ctd\u003e30-60 minutes (Viagra), 15-30 mins (Cialis)\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"2635\" data-end=\"2713\"\u003e\n\u003ctd\u003e\u003cstrong data-start=\"2637\" data-end=\"2649\"\u003eDuration\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd\u003e6-12 hours (sometimes longer)\u003c\/td\u003e\n\u003ctd\u003e4-36 hours (Cialis longest)\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"2714\" data-end=\"2762\"\u003e\n\u003ctd\u003e\u003cstrong data-start=\"2716\" data-end=\"2734\"\u003eAdministration\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd\u003eInjection\u003c\/td\u003e\n\u003ctd\u003eOral tablet\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"2763\" data-end=\"2828\"\u003e\n\u003ctd\u003e\u003cstrong data-start=\"2765\" data-end=\"2782\"\u003eUse for Women\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd\u003eYes, FDA-approved for HSDD\u003c\/td\u003e\n\u003ctd\u003eNot approved\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003c\/tbody\u003e\n\u003c\/table\u003e\n\u003c\/div\u003e\n\u003ch4 data-start=\"2830\" data-end=\"2866\"\u003e\u003cstrong data-start=\"2835\" data-end=\"2864\"\u003eLegality and Availability\u003c\/strong\u003e\u003c\/h4\u003e\n\u003cul data-start=\"2867\" data-end=\"3040\"\u003e\n\u003cli data-start=\"2867\" data-end=\"2917\"\u003e\n\u003cstrong data-start=\"2869\" data-end=\"2896\"\u003eFDA-approved as Vyleesi\u003c\/strong\u003e for HSDD in women.\u003c\/li\u003e\n\u003cli data-start=\"2918\" data-end=\"2964\"\u003eAvailable \u003cstrong data-start=\"2930\" data-end=\"2950\"\u003evia prescription\u003c\/strong\u003e in the U.S.\u003c\/li\u003e\n\u003cli data-start=\"2965\" data-end=\"3040\"\u003eOften sourced \u003cstrong data-start=\"2981\" data-end=\"2994\"\u003eoff-label\u003c\/strong\u003e from peptide vendors for research purposes\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e \u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eReferences\u003cmeta charset=\"UTF-8\"\u003e\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli data-start=\"122\" data-end=\"491\"\u003e\n\u003cp data-start=\"125\" data-end=\"305\"\u003e\u003cstrong data-start=\"125\" data-end=\"185\"\u003eiamond, L. E., Earle, D. C., Garcia, W. D., \u0026amp; Spana, C.\u003c\/strong\u003e (2006). \u003cem data-start=\"194\" data-end=\"256\"\u003eBremelanotide: An overview of preclinical and clinical data.\u003c\/em\u003e \u003cstrong data-start=\"257\" data-end=\"303\"\u003eJournal of Sexual Medicine, 3(5), 716-726.\u003c\/strong\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"493\" data-end=\"890\"\u003e\n\u003cp data-start=\"496\" data-end=\"713\"\u003e\u003cstrong data-start=\"496\" data-end=\"562\"\u003eKingsberg, S. A., Clayton, A. H., Pfaus, J. G., \u0026amp; Simon, J. A.\u003c\/strong\u003e (2019). \u003cem data-start=\"571\" data-end=\"665\"\u003eBremelanotide for the treatment of hypoactive sexual desire disorder in premenopausal women.\u003c\/em\u003e \u003cstrong data-start=\"666\" data-end=\"711\"\u003eObstetrics \u0026amp; Gynecology, 134(4), 753-765.\u003c\/strong\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"892\" data-end=\"1366\"\u003e\n\u003cp data-start=\"895\" data-end=\"1186\"\u003e\u003cstrong data-start=\"895\" data-end=\"917\"\u003eSafarinejad, M. R.\u003c\/strong\u003e (2008). \u003cem data-start=\"926\" data-end=\"1137\"\u003eEvaluation of the efficacy, safety, and characterization of intranasal bremelanotide in the treatment of erectile dysfunction: A prospective, randomized, double-blind, placebo-controlled, parallel-group trial.\u003c\/em\u003e\u003cstrong data-start=\"1138\" data-end=\"1184\"\u003eJournal of Sexual Medicine, 5(4), 866-873.\u003c\/strong\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e \u003c\/p\u003e","brand":"Mijn winkel","offers":[{"title":"Default Title","offer_id":52684862456146,"sku":"10","price":32.5,"currency_code":"EUR","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/1048\/0956\/2450\/files\/PT-141_10mg.png?v=1770834921","url":"https:\/\/sciencepeptideslab.com\/products\/pt-141-10mg-vial","provider":"Science Peptides Lab","version":"1.0","type":"link"}