{"product_id":"tbl150rad150-100x10mg-copy","title":"TBL-150(rad150) 1g","description":"\u003cp\u003e\u003cstrong\u003e\u003cspan style=\"color: rgb(255, 42, 0);\"\u003e                                                \u003cspan style=\"text-decoration: underline;\"\u003eNOT \u003c\/span\u003e\u003cspan style=\"text-decoration: underline;\"\u003eFOR HUMAN \u003c\/span\u003e\u003c\/span\u003e\u003cspan style=\"text-decoration: underline;\"\u003e\u003cspan style=\"color: rgb(255, 42, 0); text-decoration: underline;\"\u003eCONSUMPTION\u003cmeta charset=\"UTF-8\"\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp data-start=\"180\" data-end=\"700\"\u003e\u003cstrong\u003eTLB-150\u003c\/strong\u003e (RAD-150 benzoate) is an \u003cstrong data-start=\"246\" data-end=\"325\"\u003einvestigational, non-steroidal selective androgen receptor modulator (SARM)\u003c\/strong\u003e. It is widely described as the \u003cstrong data-start=\"357\" data-end=\"407\"\u003ebenzoate ester analogue of RAD-140 (testolone)\u003c\/strong\u003e, engineered to maintain \u003cstrong data-start=\"432\" data-end=\"450\"\u003eAR selectivity\u003c\/strong\u003e while potentially \u003cstrong data-start=\"469\" data-end=\"491\"\u003eextending exposure\u003c\/strong\u003e versus the parent scaffold. In vitro vendor data list potent \u003cstrong data-start=\"553\" data-end=\"570\"\u003eAR modulation\u003c\/strong\u003e in the sub-micromolar range; no approved medical indication or registrational trials exist. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003chr data-start=\"702\" data-end=\"705\"\u003e\n\u003ch3 data-start=\"707\" data-end=\"765\"\u003eAdditional Benefits of TLB-150 Now Under Investigation\u003c\/h3\u003e\n\u003cdiv class=\"_tableContainer_1rjym_1\"\u003e\n\u003cdiv class=\"_tableWrapper_1rjym_13 group flex w-fit flex-col-reverse\" tabindex=\"-1\"\u003e\n\u003ctable data-start=\"767\" data-end=\"2415\" class=\"w-fit min-w-(--thread-content-width)\"\u003e\n\u003cthead data-start=\"767\" data-end=\"795\"\u003e\n\u003ctr data-start=\"767\" data-end=\"795\"\u003e\n\u003cth data-start=\"767\" data-end=\"777\" data-col-size=\"md\"\u003eBenefit\u003c\/th\u003e\n\u003cth data-start=\"777\" data-end=\"795\" data-col-size=\"xl\"\u003eKey take-aways\u003c\/th\u003e\n\u003c\/tr\u003e\n\u003c\/thead\u003e\n\u003ctbody data-start=\"806\" data-end=\"2415\"\u003e\n\u003ctr data-start=\"806\" data-end=\"1051\"\u003e\n\u003ctd data-start=\"806\" data-end=\"845\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"808\" data-end=\"844\"\u003e1 Duration\/steadiness vs RAD-140\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"845\" data-end=\"1051\" data-col-size=\"xl\"\u003eThe \u003cstrong data-start=\"851\" data-end=\"869\"\u003ebenzoate ester\u003c\/strong\u003e is promoted to \u003cstrong data-start=\"885\" data-end=\"912\"\u003eprolong active lifespan\u003c\/strong\u003e and smooth concentration–time curves compared with RAD-140; this remains \u003cstrong data-start=\"986\" data-end=\"1010\"\u003eunverified in humans\u003c\/strong\u003e. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/sportstechnologylabs.com\/product\/rad-150\/?srsltid=AfmBOoq-zirgTA7poAH6axsdC9C-HgzbahFnFRrls6GWLOYeQzwa4mK9\u0026amp;utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/sportstechnologylabs.com\/product\/rad-150\/?srsltid=AfmBOoq-zirgTA7poAH6axsdC9C-HgzbahFnFRrls6GWLOYeQzwa4mK9\u0026amp;utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eSports Technology Labs\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\n\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"1052\" data-end=\"1266\"\u003e\n\u003ctd data-start=\"1052\" data-end=\"1092\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"1054\" data-end=\"1091\"\u003e2 Muscle anabolism (class effect)\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"1092\" data-end=\"1266\" data-col-size=\"xl\"\u003eAs an AR agonist, TLB-150 is positioned to \u003cstrong data-start=\"1137\" data-end=\"1163\"\u003eincrease fat-free mass\u003c\/strong\u003e and \u003cstrong data-start=\"1168\" data-end=\"1180\"\u003estrength\u003c\/strong\u003e similarly to first-gen SARMs—direct human efficacy data for TLB-150 are \u003cstrong data-start=\"1253\" data-end=\"1263\"\u003eabsent\u003c\/strong\u003e.\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"1267\" data-end=\"1431\"\u003e\n\u003ctd data-start=\"1267\" data-end=\"1303\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"1269\" data-end=\"1302\"\u003e3 Bone support (class effect)\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"1303\" data-end=\"1431\" data-col-size=\"xl\"\u003eSARMs up-regulate \u003cstrong data-start=\"1323\" data-end=\"1337\"\u003eosteoblast\u003c\/strong\u003e pathways and improve BMD in animals; TLB-150 is presumed comparable pending direct studies.\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"1432\" data-end=\"1569\"\u003e\n\u003ctd data-start=\"1432\" data-end=\"1457\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"1434\" data-end=\"1456\"\u003e4 Oral convenience\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"1457\" data-end=\"1569\" data-col-size=\"xl\"\u003e\n\u003cstrong data-start=\"1459\" data-end=\"1478\"\u003eOnce-daily oral\u003c\/strong\u003e SARM paradigms favor adherence vs injectables; specific TLB-150 PK in humans is unknown.\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"1570\" data-end=\"1775\"\u003e\n\u003ctd data-start=\"1570\" data-end=\"1617\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"1572\" data-end=\"1616\"\u003e5 Potentially lower androgenic “baggage”\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"1617\" data-end=\"1775\" data-col-size=\"xl\"\u003eLike other non-steroidal SARMs, design intent is \u003cstrong data-start=\"1668\" data-end=\"1695\"\u003emuscle\/bone selectivity\u003c\/strong\u003e with \u003cstrong data-start=\"1701\" data-end=\"1735\"\u003eless prostate\/skin stimulation\u003c\/strong\u003e than testosterone—needs confirmation.\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"1776\" data-end=\"1935\"\u003e\n\u003ctd data-start=\"1776\" data-end=\"1809\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"1778\" data-end=\"1808\"\u003e6 Research-use positioning\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"1809\" data-end=\"1935\" data-col-size=\"xl\"\u003eCommercial listings emphasize \u003cstrong data-start=\"1841\" data-end=\"1862\"\u003eresearch-use only\u003c\/strong\u003e and lack of regulatory approval. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.medchemexpress.com\/tlb-150-benzoate.html?srsltid=AfmBOoqt13PcEDRA5-7IsN4TnsCNlIyBV8fv-HwVzrzjcAKwa6Hph5hF\u0026amp;utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.medchemexpress.com\/tlb-150-benzoate.html?srsltid=AfmBOoqt13PcEDRA5-7IsN4TnsCNlIyBV8fv-HwVzrzjcAKwa6Hph5hF\u0026amp;utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003emedchemexpress.com\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\n\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"1936\" data-end=\"2092\"\u003e\n\u003ctd data-start=\"1936\" data-end=\"1988\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"1938\" data-end=\"1987\"\u003e7 SARM-class synergy with resistance training\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"1988\" data-end=\"2092\" data-col-size=\"xl\"\u003eExpect \u003cstrong data-start=\"1997\" data-end=\"2011\"\u003eadditivity\u003c\/strong\u003e with structured training\/protein adequacy (extrapolated from SARM literature).\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"2093\" data-end=\"2255\"\u003e\n\u003ctd data-start=\"2093\" data-end=\"2120\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"2095\" data-end=\"2119\"\u003e8 Dosing flexibility\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"2120\" data-end=\"2255\" data-col-size=\"xl\"\u003eIf ester prolongation holds, \u003cstrong data-start=\"2151\" data-end=\"2172\"\u003elower\/fewer doses\u003c\/strong\u003e could yield similar exposure (hypothesis). \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/sportstechnologylabs.com\/product\/rad-150\/?srsltid=AfmBOoq-zirgTA7poAH6axsdC9C-HgzbahFnFRrls6GWLOYeQzwa4mK9\u0026amp;utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/sportstechnologylabs.com\/product\/rad-150\/?srsltid=AfmBOoq-zirgTA7poAH6axsdC9C-HgzbahFnFRrls6GWLOYeQzwa4mK9\u0026amp;utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eSports Technology Labs\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\n\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"2256\" data-end=\"2415\"\u003e\n\u003ctd data-start=\"2256\" data-end=\"2281\" data-col-size=\"md\"\u003e\u003cstrong data-start=\"2258\" data-end=\"2280\"\u003e9 Doping relevance\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-start=\"2281\" data-end=\"2415\" data-col-size=\"xl\"\u003eAs a SARM, TLB-150 would be \u003cstrong data-start=\"2311\" data-end=\"2338\"\u003eprohibited at all times\u003c\/strong\u003e under \u003cstrong data-start=\"2345\" data-end=\"2374\"\u003eWADA S1 (Anabolic Agents)\u003c\/strong\u003e. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.usada.org\/spirit-of-sport\/selective-androgen-receptor-modulators-sarms-prohibited-class-anabolic-agents\/?utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.usada.org\/spirit-of-sport\/selective-androgen-receptor-modulators-sarms-prohibited-class-anabolic-agents\/?utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eU.S. Anti-Doping Agency (USADA)\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.wada-ama.org\/en\/prohibited-list?utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.wada-ama.org\/en\/prohibited-list?utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003ewada-ama.org\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\n\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003c\/tbody\u003e\n\u003c\/table\u003e\n\u003c\/div\u003e\n\u003c\/div\u003e\n\u003chr data-start=\"2417\" data-end=\"2420\"\u003e\n\u003ch2 data-start=\"2422\" data-end=\"2457\"\u003e2. Molecular Mechanism of Action\u003c\/h2\u003e\n\u003ch3 data-start=\"2459\" data-end=\"2494\"\u003e2.1 Receptor Pharmacodynamics\u003c\/h3\u003e\n\u003cp data-start=\"2495\" data-end=\"2820\"\u003eTLB-150 binds the \u003cstrong data-start=\"2513\" data-end=\"2539\"\u003eandrogen receptor (AR)\u003c\/strong\u003e, promoting \u003cstrong data-start=\"2551\" data-end=\"2576\"\u003enuclear translocation\u003c\/strong\u003e and \u003cstrong data-start=\"2581\" data-end=\"2609\"\u003eARE-driven transcription\u003c\/strong\u003e. In muscle, AR activation up-regulates \u003cstrong data-start=\"2649\" data-end=\"2661\"\u003emTOR\/S6K\u003c\/strong\u003e and suppresses \u003cstrong data-start=\"2677\" data-end=\"2690\"\u003eatrogenes\u003c\/strong\u003e (MAFbx\/MuRF1); in bone, AR signaling supports \u003cstrong data-start=\"2737\" data-end=\"2759\"\u003eosteoblastogenesis\u003c\/strong\u003e and trabecular integrity (inferred from SARM class biology).\u003c\/p\u003e\n\u003ch3 data-start=\"2822\" data-end=\"2849\"\u003e2.2 Down-stream Biology\u003c\/h3\u003e\n\u003cdiv class=\"_tableContainer_1rjym_1\"\u003e\n\u003cdiv class=\"_tableWrapper_1rjym_13 group flex w-fit flex-col-reverse\" tabindex=\"-1\"\u003e\n\u003ctable data-start=\"2851\" data-end=\"3224\" class=\"w-fit min-w-(--thread-content-width)\"\u003e\n\u003cthead data-start=\"2851\" data-end=\"2893\"\u003e\n\u003ctr data-start=\"2851\" data-end=\"2893\"\u003e\n\u003cth data-start=\"2851\" data-end=\"2861\" data-col-size=\"sm\"\u003ePathway\u003c\/th\u003e\n\u003cth data-start=\"2861\" data-end=\"2882\" data-col-size=\"md\"\u003eFunctional outcome\u003c\/th\u003e\n\u003cth data-start=\"2882\" data-end=\"2893\" data-col-size=\"sm\"\u003eContext\u003c\/th\u003e\n\u003c\/tr\u003e\n\u003c\/thead\u003e\n\u003ctbody data-start=\"2908\" data-end=\"3224\"\u003e\n\u003ctr data-start=\"2908\" data-end=\"2994\"\u003e\n\u003ctd data-start=\"2908\" data-end=\"2931\" data-col-size=\"sm\"\u003eAR → mTOR\/S6K\/4E-BP1\u003c\/td\u003e\n\u003ctd data-start=\"2931\" data-end=\"2975\" data-col-size=\"md\"\u003e↑ Protein synthesis, myofiber hypertrophy\u003c\/td\u003e\n\u003ctd data-start=\"2975\" data-end=\"2994\" data-col-size=\"sm\"\u003eSkeletal muscle\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"2995\" data-end=\"3063\"\u003e\n\u003ctd data-start=\"2995\" data-end=\"3024\" data-col-size=\"sm\"\u003eAR ↔ Wnt\/β-catenin\/Osterix\u003c\/td\u003e\n\u003ctd data-col-size=\"md\" data-start=\"3024\" data-end=\"3055\"\u003e↑ Osteoblast activity, ↑ BMD\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"3055\" data-end=\"3063\"\u003eBone\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"3064\" data-end=\"3144\"\u003e\n\u003ctd data-start=\"3064\" data-end=\"3091\" data-col-size=\"sm\"\u003e↓ FoxO\/ubiquitin ligases\u003c\/td\u003e\n\u003ctd data-col-size=\"md\" data-start=\"3091\" data-end=\"3124\"\u003e↓ Proteolysis (anti-catabolic)\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"3124\" data-end=\"3144\"\u003eCatabolic stress\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"3145\" data-end=\"3224\"\u003e\n\u003ctd data-start=\"3145\" data-end=\"3165\" data-col-size=\"sm\"\u003eHPG-axis feedback\u003c\/td\u003e\n\u003ctd data-col-size=\"md\" data-start=\"3165\" data-end=\"3203\"\u003e↓ LH\/FSH\/testosterone (suppression)\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"3203\" data-end=\"3224\"\u003ePituitary–gonadal\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003c\/tbody\u003e\n\u003c\/table\u003e\n\u003c\/div\u003e\n\u003c\/div\u003e\n\u003chr data-start=\"3226\" data-end=\"3229\"\u003e\n\u003ch2 data-start=\"3231\" data-end=\"3253\"\u003e3. Pharmacokinetics\u003c\/h2\u003e\n\u003cul data-start=\"3255\" data-end=\"3766\"\u003e\n\u003cli data-start=\"3255\" data-end=\"3290\"\u003e\n\u003cp data-start=\"3257\" data-end=\"3290\"\u003e\u003cstrong data-start=\"3257\" data-end=\"3267\"\u003eRoute:\u003c\/strong\u003e Oral (research use).\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"3291\" data-end=\"3495\"\u003e\n\u003cp data-start=\"3293\" data-end=\"3495\"\u003e\u003cstrong data-start=\"3293\" data-end=\"3314\"\u003eDesign rationale:\u003c\/strong\u003e \u003cstrong data-start=\"3315\" data-end=\"3342\"\u003eBenzoate esterification\u003c\/strong\u003e of RAD-140 intended to \u003cstrong data-start=\"3366\" data-end=\"3411\"\u003eenhance stability and effective half-life\u003c\/strong\u003e; quantitative human PK is \u003cstrong data-start=\"3438\" data-end=\"3454\"\u003eundetermined\u003c\/strong\u003e. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/sportstechnologylabs.com\/product\/rad-150\/?srsltid=AfmBOoq-zirgTA7poAH6axsdC9C-HgzbahFnFRrls6GWLOYeQzwa4mK9\u0026amp;utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/sportstechnologylabs.com\/product\/rad-150\/?srsltid=AfmBOoq-zirgTA7poAH6axsdC9C-HgzbahFnFRrls6GWLOYeQzwa4mK9\u0026amp;utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eSports Technology Labs\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"3496\" data-end=\"3642\"\u003e\n\u003cp data-start=\"3498\" data-end=\"3642\"\u003e\u003cstrong data-start=\"3498\" data-end=\"3523\"\u003eMetabolism\/clearance:\u003c\/strong\u003e Expected \u003cstrong data-start=\"3533\" data-end=\"3553\"\u003eester hydrolysis\u003c\/strong\u003e → RAD-140-like core + oxidative\/conjugative metabolism; formal human data unavailable.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"3643\" data-end=\"3766\"\u003e\n\u003cp data-start=\"3645\" data-end=\"3766\"\u003e\u003cstrong data-start=\"3645\" data-end=\"3659\"\u003eDetection:\u003c\/strong\u003e As a SARM, long-term metabolites may extend detection windows in doping control (extrapolated from class).\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003chr data-start=\"3768\" data-end=\"3771\"\u003e\n\u003ch2 data-start=\"3773\" data-end=\"3818\"\u003e4. Pre-clinical and Translational Evidence\u003c\/h2\u003e\n\u003ch3 data-start=\"3820\" data-end=\"3859\"\u003e4.1 Identity \u0026amp; in-vitro profiling\u003c\/h3\u003e\n\u003cp data-start=\"3860\" data-end=\"4090\"\u003eCommercial technical sheets list \u003cstrong data-start=\"3893\" data-end=\"3910\"\u003eAR modulation\u003c\/strong\u003e with \u003cstrong data-start=\"3916\" data-end=\"3934\"\u003esub-µM potency\u003c\/strong\u003e and \u003cstrong data-start=\"3939\" data-end=\"3959\"\u003eCAS 1208070-53-4\u003c\/strong\u003e; peer-reviewed \u003cstrong data-start=\"3975\" data-end=\"3986\"\u003ein-vivo\u003c\/strong\u003eefficacy for TLB-150 specifically is \u003cstrong data-start=\"4024\" data-end=\"4051\"\u003elimited\/publicly sparse\u003c\/strong\u003e. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.medchemexpress.com\/tlb-150-benzoate.html?srsltid=AfmBOoqt13PcEDRA5-7IsN4TnsCNlIyBV8fv-HwVzrzjcAKwa6Hph5hF\u0026amp;utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.medchemexpress.com\/tlb-150-benzoate.html?srsltid=AfmBOoqt13PcEDRA5-7IsN4TnsCNlIyBV8fv-HwVzrzjcAKwa6Hph5hF\u0026amp;utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003emedchemexpress.com\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003ch3 data-start=\"4092\" data-end=\"4144\"\u003e4.2 Extrapolation from RAD-140\/SARM literature\u003c\/h3\u003e\n\u003cp data-start=\"4145\" data-end=\"4357\"\u003eAnabolic \u003cstrong data-start=\"4154\" data-end=\"4167\"\u003eFFM gains\u003c\/strong\u003e, \u003cstrong data-start=\"4169\" data-end=\"4194\"\u003estrength improvements\u003c\/strong\u003e, and \u003cstrong data-start=\"4200\" data-end=\"4219\"\u003ebone protection\u003c\/strong\u003e are well described for earlier SARMs in animals and small human studies; whether \u003cstrong data-start=\"4301\" data-end=\"4312\"\u003eTLB-150\u003c\/strong\u003e surpasses RAD-140 clinically is \u003cstrong data-start=\"4345\" data-end=\"4356\"\u003eunknown\u003c\/strong\u003e.\u003c\/p\u003e\n\u003cblockquote data-start=\"4359\" data-end=\"4503\"\u003e\n\u003cp data-start=\"4361\" data-end=\"4503\"\u003e\u003cstrong data-start=\"4361\" data-end=\"4387\"\u003eEvidence quality note:\u003c\/strong\u003e TLB-150 data are \u003cstrong data-start=\"4405\" data-end=\"4446\"\u003elargely vendor-level and pre-clinical\u003c\/strong\u003e; there are \u003cstrong data-start=\"4458\" data-end=\"4489\"\u003eno authoritative human RCTs\u003c\/strong\u003e or approvals.\u003c\/p\u003e\n\u003c\/blockquote\u003e\n\u003chr data-start=\"4505\" data-end=\"4508\"\u003e\n\u003ch2 data-start=\"4510\" data-end=\"4543\"\u003e5. Emerging Clinical Interests\u003c\/h2\u003e\n\u003cdiv class=\"_tableContainer_1rjym_1\"\u003e\n\u003cdiv class=\"_tableWrapper_1rjym_13 group flex w-fit flex-col-reverse\" tabindex=\"-1\"\u003e\n\u003ctable data-start=\"4545\" data-end=\"5040\" class=\"w-fit min-w-(--thread-content-width)\"\u003e\n\u003cthead data-start=\"4545\" data-end=\"4583\"\u003e\n\u003ctr data-start=\"4545\" data-end=\"4583\"\u003e\n\u003cth data-start=\"4545\" data-end=\"4553\" data-col-size=\"sm\"\u003eField\u003c\/th\u003e\n\u003cth data-start=\"4553\" data-end=\"4565\" data-col-size=\"md\"\u003eRationale\u003c\/th\u003e\n\u003cth data-start=\"4565\" data-end=\"4583\" data-col-size=\"sm\"\u003eCurrent status\u003c\/th\u003e\n\u003c\/tr\u003e\n\u003c\/thead\u003e\n\u003ctbody data-start=\"4598\" data-end=\"5040\"\u003e\n\u003ctr data-start=\"4598\" data-end=\"4692\"\u003e\n\u003ctd data-start=\"4598\" data-end=\"4621\" data-col-size=\"sm\"\u003e\u003cstrong data-start=\"4600\" data-end=\"4620\"\u003eSarcopenia\/rehab\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-col-size=\"md\" data-start=\"4621\" data-end=\"4667\"\u003eOral anabolic with putative longer exposure\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"4667\" data-end=\"4692\"\u003eConcept\/extrapolation\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"4693\" data-end=\"4771\"\u003e\n\u003ctd data-start=\"4693\" data-end=\"4710\" data-col-size=\"sm\"\u003e\u003cstrong data-start=\"4695\" data-end=\"4709\"\u003eOsteopenia\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-col-size=\"md\" data-start=\"4710\" data-end=\"4745\"\u003eBone-anabolic SARM class biology\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"4745\" data-end=\"4771\"\u003ePre-clinical rationale\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"4772\" data-end=\"4898\"\u003e\n\u003ctd data-start=\"4772\" data-end=\"4806\" data-col-size=\"sm\"\u003e\u003cstrong data-start=\"4774\" data-end=\"4805\"\u003eMale contraception research\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-col-size=\"md\" data-start=\"4806\" data-end=\"4879\"\u003eStrong HPG suppression is a SARM class effect—\u003cstrong data-start=\"4854\" data-end=\"4866\"\u003eunproven\u003c\/strong\u003e for TLB-150\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"4879\" data-end=\"4898\"\u003eHypothesis only\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"4899\" data-end=\"5040\"\u003e\n\u003ctd data-start=\"4899\" data-end=\"4929\" data-col-size=\"sm\"\u003e\u003cstrong data-start=\"4901\" data-end=\"4928\"\u003eAthletics (illicit use)\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-col-size=\"md\" data-start=\"4929\" data-end=\"4979\"\u003eOral potency + duration = high misuse potential\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"4979\" data-end=\"5040\"\u003e\n\u003cstrong data-start=\"4981\" data-end=\"5000\"\u003eWADA-prohibited\u003c\/strong\u003e \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.usada.org\/spirit-of-sport\/selective-androgen-receptor-modulators-sarms-prohibited-class-anabolic-agents\/?utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.usada.org\/spirit-of-sport\/selective-androgen-receptor-modulators-sarms-prohibited-class-anabolic-agents\/?utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eU.S. Anti-Doping Agency (USADA)\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\n\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003c\/tbody\u003e\n\u003c\/table\u003e\n\u003c\/div\u003e\n\u003c\/div\u003e\n\u003chr data-start=\"5042\" data-end=\"5045\"\u003e\n\u003ch2 data-start=\"5047\" data-end=\"5076\"\u003e6. Safety and Tolerability\u003c\/h2\u003e\n\u003cul data-start=\"5078\" data-end=\"5680\"\u003e\n\u003cli data-start=\"5078\" data-end=\"5298\"\u003e\n\u003cp data-start=\"5080\" data-end=\"5298\"\u003e\u003cstrong data-start=\"5080\" data-end=\"5113\"\u003eKnown\/expected class effects:\u003c\/strong\u003e\u003cbr data-start=\"5113\" data-end=\"5116\"\u003e\u003cstrong data-start=\"5118\" data-end=\"5142\"\u003eHPG-axis suppression\u003c\/strong\u003e (↓ LH\/FSH\/testosterone), \u003cstrong data-start=\"5168\" data-end=\"5187\"\u003eHDL-C reduction\u003c\/strong\u003e (± ↑ LDL\/TG), possible \u003cstrong data-start=\"5211\" data-end=\"5233\"\u003eALT\/AST elevations\u003c\/strong\u003e, \u003cstrong data-start=\"5235\" data-end=\"5253\"\u003eacne\/oily skin\u003c\/strong\u003e, \u003cstrong data-start=\"5255\" data-end=\"5272\"\u003emood\/insomnia\u003c\/strong\u003e, \u003cstrong data-start=\"5274\" data-end=\"5295\"\u003emild ↑ hematocrit\u003c\/strong\u003e.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"5299\" data-end=\"5426\"\u003e\n\u003cp data-start=\"5301\" data-end=\"5426\"\u003e\u003cstrong data-start=\"5301\" data-end=\"5326\"\u003eUnknowns for TLB-150:\u003c\/strong\u003e \u003cstrong data-start=\"5327\" data-end=\"5339\"\u003eHuman PK\u003c\/strong\u003e, \u003cstrong data-start=\"5341\" data-end=\"5358\"\u003edose–response\u003c\/strong\u003e, \u003cstrong data-start=\"5360\" data-end=\"5393\"\u003elong-term hepatic\/CV outcomes\u003c\/strong\u003e, \u003cstrong data-start=\"5395\" data-end=\"5415\"\u003eneuropsychiatric\u003c\/strong\u003esignals.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"5427\" data-end=\"5535\"\u003e\n\u003cp data-start=\"5429\" data-end=\"5535\"\u003e\u003cstrong data-start=\"5429\" data-end=\"5447\"\u003eQuality risks:\u003c\/strong\u003e Grey-market products show \u003cstrong data-start=\"5474\" data-end=\"5502\"\u003eadulteration\/mislabeling\u003c\/strong\u003e; use outside trials is unsafe.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"5536\" data-end=\"5623\"\u003e\n\u003cp data-start=\"5538\" data-end=\"5623\"\u003e\u003cstrong data-start=\"5538\" data-end=\"5560\"\u003eDrug interactions:\u003c\/strong\u003e Potential hepatic enzyme interactions (class consideration).\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"5624\" data-end=\"5680\"\u003e\n\u003cp data-start=\"5626\" data-end=\"5680\"\u003e\u003cstrong data-start=\"5626\" data-end=\"5640\"\u003ePregnancy:\u003c\/strong\u003e Contraindicated (androgenic mechanism).\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp data-start=\"5682\" data-end=\"5711\"\u003e\u003cstrong data-start=\"5682\" data-end=\"5711\"\u003eComparative safety matrix\u003c\/strong\u003e\u003c\/p\u003e\n\u003cdiv class=\"_tableContainer_1rjym_1\"\u003e\n\u003cdiv class=\"_tableWrapper_1rjym_13 group flex w-fit flex-col-reverse\" tabindex=\"-1\"\u003e\n\u003ctable data-start=\"5713\" data-end=\"6192\" class=\"w-fit min-w-(--thread-content-width)\"\u003e\n\u003cthead data-start=\"5713\" data-end=\"5800\"\u003e\n\u003ctr data-start=\"5713\" data-end=\"5800\"\u003e\n\u003cth data-start=\"5713\" data-end=\"5723\" data-col-size=\"sm\"\u003eConcern\u003c\/th\u003e\n\u003cth data-start=\"5723\" data-end=\"5747\" data-col-size=\"sm\"\u003e\u003cstrong data-start=\"5725\" data-end=\"5746\"\u003eTLB-150 (RAD-150)\u003c\/strong\u003e\u003c\/th\u003e\n\u003cth data-start=\"5747\" data-end=\"5773\" data-col-size=\"sm\"\u003e\u003cstrong data-start=\"5749\" data-end=\"5772\"\u003eRAD-140 (testolone)\u003c\/strong\u003e\u003c\/th\u003e\n\u003cth data-start=\"5773\" data-end=\"5800\" data-col-size=\"sm\"\u003e\u003cstrong data-start=\"5775\" data-end=\"5798\"\u003eEnobosarm (MK-2866)\u003c\/strong\u003e\u003c\/th\u003e\n\u003c\/tr\u003e\n\u003c\/thead\u003e\n\u003ctbody data-start=\"5819\" data-end=\"6192\"\u003e\n\u003ctr data-start=\"5819\" data-end=\"5940\"\u003e\n\u003ctd data-start=\"5819\" data-end=\"5834\" data-col-size=\"sm\"\u003eOral potency\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"5834\" data-end=\"5867\"\u003ePresumed \u003cstrong data-start=\"5845\" data-end=\"5853\"\u003ehigh\u003c\/strong\u003e (unverified)\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"5867\" data-end=\"5903\"\u003e\n\u003cstrong data-start=\"5869\" data-end=\"5877\"\u003eHigh\u003c\/strong\u003e (preclinical + forensic)\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"5903\" data-end=\"5940\"\u003e\n\u003cstrong data-start=\"5905\" data-end=\"5922\"\u003eModerate–high\u003c\/strong\u003e (human Phase 2)\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"5941\" data-end=\"6010\"\u003e\n\u003ctd data-start=\"5941\" data-end=\"5952\" data-col-size=\"sm\"\u003eDuration\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"5952\" data-end=\"5982\"\u003e\n\u003cstrong data-start=\"5954\" data-end=\"5973\"\u003eDesigned longer\u003c\/strong\u003e (ester)\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"5982\" data-end=\"6001\"\u003eShorter vs ester\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6001\" data-end=\"6010\"\u003e~24 h\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"6011\" data-end=\"6092\"\u003e\n\u003ctd data-start=\"6011\" data-end=\"6024\" data-col-size=\"sm\"\u003eHuman data\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6024\" data-end=\"6048\"\u003e\u003cstrong data-start=\"6026\" data-end=\"6047\"\u003eNone\/very limited\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6048\" data-end=\"6072\"\u003eLimited (non-pivotal)\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6072\" data-end=\"6092\"\u003ePhase 2 datasets\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"6093\" data-end=\"6132\"\u003e\n\u003ctd data-start=\"6093\" data-end=\"6106\" data-col-size=\"sm\"\u003eHDL impact\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6106\" data-end=\"6123\"\u003eExpected \u003cstrong data-start=\"6117\" data-end=\"6122\"\u003e↓\u003c\/strong\u003e\n\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6123\" data-end=\"6127\"\u003e↓\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6127\" data-end=\"6132\"\u003e↓\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003ctr data-start=\"6133\" data-end=\"6192\"\u003e\n\u003ctd data-start=\"6133\" data-end=\"6151\" data-col-size=\"sm\"\u003eHPG suppression\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6151\" data-end=\"6171\"\u003e\u003cstrong data-start=\"6153\" data-end=\"6170\"\u003eLikely strong\u003c\/strong\u003e\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6171\" data-end=\"6180\"\u003eStrong\u003c\/td\u003e\n\u003ctd data-col-size=\"sm\" data-start=\"6180\" data-end=\"6192\"\u003eModerate\u003c\/td\u003e\n\u003c\/tr\u003e\n\u003c\/tbody\u003e\n\u003c\/table\u003e\n\u003c\/div\u003e\n\u003c\/div\u003e\n\u003chr data-start=\"6194\" data-end=\"6197\"\u003e\n\u003ch2 data-start=\"6199\" data-end=\"6225\"\u003e7. Regulatory Landscape\u003c\/h2\u003e\n\u003cul data-start=\"6227\" data-end=\"6518\"\u003e\n\u003cli data-start=\"6227\" data-end=\"6348\"\u003e\n\u003cp data-start=\"6229\" data-end=\"6348\"\u003e\u003cstrong data-start=\"6229\" data-end=\"6243\"\u003eApprovals:\u003c\/strong\u003e \u003cstrong data-start=\"6244\" data-end=\"6252\"\u003eNone\u003c\/strong\u003e; marketed as \u003cstrong data-start=\"6266\" data-end=\"6287\"\u003eresearch-use only\u003c\/strong\u003e by chemical vendors. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.medchemexpress.com\/tlb-150-benzoate.html?srsltid=AfmBOoqt13PcEDRA5-7IsN4TnsCNlIyBV8fv-HwVzrzjcAKwa6Hph5hF\u0026amp;utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.medchemexpress.com\/tlb-150-benzoate.html?srsltid=AfmBOoqt13PcEDRA5-7IsN4TnsCNlIyBV8fv-HwVzrzjcAKwa6Hph5hF\u0026amp;utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003emedchemexpress.com\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"6349\" data-end=\"6518\"\u003e\n\u003cp data-start=\"6351\" data-end=\"6518\"\u003e\u003cstrong data-start=\"6351\" data-end=\"6361\"\u003eSport:\u003c\/strong\u003e \u003cstrong data-start=\"6362\" data-end=\"6390\"\u003eAll SARMs are prohibited\u003c\/strong\u003e at all times under \u003cstrong data-start=\"6410\" data-end=\"6421\"\u003eWADA S1\u003c\/strong\u003e; athletes face sanction even for contaminated supplements. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.usada.org\/spirit-of-sport\/selective-androgen-receptor-modulators-sarms-prohibited-class-anabolic-agents\/?utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.usada.org\/spirit-of-sport\/selective-androgen-receptor-modulators-sarms-prohibited-class-anabolic-agents\/?utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eU.S. Anti-Doping Agency (USADA)\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.wada-ama.org\/en\/prohibited-list?utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.wada-ama.org\/en\/prohibited-list?utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003ewada-ama.org\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003chr data-start=\"6520\" data-end=\"6523\"\u003e\n\u003ch2 data-start=\"6525\" data-end=\"6548\"\u003e8. Future Directions\u003c\/h2\u003e\n\u003cul data-start=\"6550\" data-end=\"7072\"\u003e\n\u003cli data-start=\"6550\" data-end=\"6678\"\u003e\n\u003cp data-start=\"6552\" data-end=\"6678\"\u003e\u003cstrong data-start=\"6552\" data-end=\"6571\"\u003eAuthentic PK\/PD\u003c\/strong\u003e: First-in-human \u003cstrong data-start=\"6588\" data-end=\"6595\"\u003eGMP\u003c\/strong\u003e studies to define \u003cstrong data-start=\"6614\" data-end=\"6652\"\u003ehalf-life, exposure, metabolite ID\u003c\/strong\u003e, and \u003cstrong data-start=\"6658\" data-end=\"6675\"\u003edose–response\u003c\/strong\u003e.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"6679\" data-end=\"6784\"\u003e\n\u003cp data-start=\"6681\" data-end=\"6784\"\u003e\u003cstrong data-start=\"6681\" data-end=\"6708\"\u003eHead-to-head vs RAD-140\u003c\/strong\u003e: Demonstrate \u003cstrong data-start=\"6722\" data-end=\"6764\"\u003esuperiority (duration\/efficacy\/safety)\u003c\/strong\u003e, not just parity.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"6785\" data-end=\"6887\"\u003e\n\u003cp data-start=\"6787\" data-end=\"6887\"\u003e\u003cstrong data-start=\"6787\" data-end=\"6807\"\u003eLong-term safety\u003c\/strong\u003e: \u003cstrong data-start=\"6809\" data-end=\"6822\"\u003eLipids\/CV\u003c\/strong\u003e, \u003cstrong data-start=\"6824\" data-end=\"6835\"\u003ehepatic\u003c\/strong\u003e, \u003cstrong data-start=\"6837\" data-end=\"6859\"\u003eendocrine recovery\u003c\/strong\u003e; standardized monitoring.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"6888\" data-end=\"6957\"\u003e\n\u003cp data-start=\"6890\" data-end=\"6957\"\u003e\u003cstrong data-start=\"6890\" data-end=\"6908\"\u003eDoping science\u003c\/strong\u003e: Metabolite mapping and \u003cstrong data-start=\"6933\" data-end=\"6954\"\u003edetection windows\u003c\/strong\u003e.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"6958\" data-end=\"7072\"\u003e\n\u003cp data-start=\"6960\" data-end=\"7072\"\u003e\u003cstrong data-start=\"6960\" data-end=\"6983\"\u003eMedicinal chemistry\u003c\/strong\u003e: Optimize \u003cstrong data-start=\"6994\" data-end=\"7014\"\u003elipid neutrality\u003c\/strong\u003e and \u003cstrong data-start=\"7019\" data-end=\"7046\"\u003ereduced HPG suppression\u003c\/strong\u003e without losing anabolism.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003chr data-start=\"7074\" data-end=\"7077\"\u003e\n\u003ch3 data-start=\"7079\" data-end=\"7102\"\u003eSelected References\u003c\/h3\u003e\n\u003cul data-start=\"7104\" data-end=\"7657\"\u003e\n\u003cli data-start=\"7104\" data-end=\"7264\"\u003e\n\u003cp data-start=\"7106\" data-end=\"7264\"\u003eMedChemExpress technical page: \u003cstrong data-start=\"7137\" data-end=\"7222\"\u003e“TLB-150 Benzoate (RAD-150) — AR modulator; CAS 1208070-53-4; research-use only.”\u003c\/strong\u003e \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.medchemexpress.com\/tlb-150-benzoate.html?srsltid=AfmBOoqt13PcEDRA5-7IsN4TnsCNlIyBV8fv-HwVzrzjcAKwa6Hph5hF\u0026amp;utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.medchemexpress.com\/tlb-150-benzoate.html?srsltid=AfmBOoqt13PcEDRA5-7IsN4TnsCNlIyBV8fv-HwVzrzjcAKwa6Hph5hF\u0026amp;utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003emedchemexpress.com\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"7265\" data-end=\"7428\"\u003e\n\u003cp data-start=\"7267\" data-end=\"7428\"\u003eVendor\/scientific summaries describing \u003cstrong data-start=\"7306\" data-end=\"7350\"\u003eRAD-150 as the benzoate ester of RAD-140\u003c\/strong\u003e with \u003cstrong data-start=\"7356\" data-end=\"7385\"\u003eprolonged activity claims\u003c\/strong\u003e. \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/sportstechnologylabs.com\/product\/rad-150\/?srsltid=AfmBOoq-zirgTA7poAH6axsdC9C-HgzbahFnFRrls6GWLOYeQzwa4mK9\u0026amp;utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/sportstechnologylabs.com\/product\/rad-150\/?srsltid=AfmBOoq-zirgTA7poAH6axsdC9C-HgzbahFnFRrls6GWLOYeQzwa4mK9\u0026amp;utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eSports Technology Labs\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/lawlesslabsusa.com\/products\/tlb-150-rad150?utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/lawlesslabsusa.com\/products\/tlb-150-rad150?utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eLawless Labs USA\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"7429\" data-end=\"7557\"\u003e\n\u003cp data-start=\"7431\" data-end=\"7557\"\u003e\u003cstrong data-start=\"7431\" data-end=\"7440\"\u003eUSADA\u003c\/strong\u003e: “\u003cstrong data-start=\"7443\" data-end=\"7484\"\u003eAll SARMs are prohibited at all times\u003c\/strong\u003e (S1 ‘Other Anabolic Agents’).” \u003cspan class=\"\" data-state=\"closed\"\u003e\u003cspan class=\"ms-1 inline-flex max-w-full items-center relative top-[-0.094rem] animate-[show_150ms_ease-in]\" data-testid=\"webpage-citation-pill\"\u003e\u003ca href=\"https:\/\/www.usada.org\/spirit-of-sport\/selective-androgen-receptor-modulators-sarms-prohibited-class-anabolic-agents\/?utm_source=chatgpt.com\" rel=\"noopener\" alt=\"https:\/\/www.usada.org\/spirit-of-sport\/selective-androgen-receptor-modulators-sarms-prohibited-class-anabolic-agents\/?utm_source=chatgpt.com\" class=\"flex h-4.5 overflow-hidden rounded-xl px-2 text-[9px] font-medium text-token-text-secondary! bg-[#F4F4F4]! dark:bg-[#303030]! transition-colors duration-150 ease-in-out\" target=\"_blank\"\u003e\u003cspan class=\"relative start-0 bottom-0 flex h-full w-full items-center\"\u003e\u003cspan class=\"flex h-4 w-full items-center justify-between overflow-hidden\"\u003e\u003cspan class=\"max-w-full grow truncate overflow-hidden text-center\"\u003eU.S. Anti-Doping Agency (USADA)\u003c\/span\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/a\u003e\u003c\/span\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli data-start=\"7558\" data-end=\"7657\"\u003e\n\u003cp data-start=\"7560\" data-end=\"7657\"\u003e\u003cstrong data-start=\"7560\" data-end=\"7591\"\u003eWADA Prohibited List (2025)\u003c\/strong\u003e — International Standard.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e \u003c\/p\u003e","brand":"Mijn winkel","offers":[{"title":"Default Title","offer_id":52684848431442,"sku":"10","price":77.5,"currency_code":"EUR","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/1048\/0956\/2450\/files\/rad150_1g.png?v=1770834831","url":"https:\/\/sciencepeptideslab.com\/products\/tbl150rad150-100x10mg-copy","provider":"Science Peptides Lab","version":"1.0","type":"link"}